Catalogue number: R139300
Chemical name: Rebastinib
Synonyms: DCC-2036; DP 1919; 4-[4-[(5-tert-Butyl-2-quinolin-6-ylpyrazol-3-yl)carbamoylamino]-3-fluorophenoxy]-N-methylpyridine-2-carboxamide
CAS Number: 1020172-07-9
Possible CAS #: NA
Molecular form.: C₃₀H₂₈FN₇O₃
Appearance: Off-White Solid
Melting Point: >181°C (dec.)
Mol. Weight: 553.59
Storage: -20°C Freezer
Solubility: Methanol (Slightly)
Stability: No Data Available
Category: No Data Available
Boiling Point: No Data Available
Applications: Rebastinib shows the selectivity for growth inhibition of Bcr-Abl-positive cells by its marked inhibition of CML cell lines compared to non-CML leukemia lines. Rebastinib (DCC-2036) is a conformational control Bcr-Abl inhibitor for Abl1(WT) and Abl1(T315I) with IC50 of 0.8 nM and 4 nM, also inhibits SRC, LYN, FGR, HCK, KDR, FLT3, and Tie-2, and low activity to seen towards c-Kit. Phase 1.
Dangerous Goods Info: NA
Peer Review Product Citations:
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  Pack size Price(USD)
1mg $145.00
10mg $450.00
  Pack size Price(USD)
2.5mg $330.00
25mg $675.00

Exact Weight Packaging ($75(USD) / Vial)
Inventory Status:   In Stock

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