K162500 Chemical Structure

All Products are stable to be shipped at room temperature, unless otherwise specified.
Pack SizeQuantityPrice (USD)Sub Total
1mg
$ 45.000.0
5mg
$ 90.000.0
10mg
$ 125.000.0
25mg
$ 305.000.0
50mg
$ 580.000.0
100mg
$ 1010.000.0
Exact Weight Packaging
$ 95.000.0
Total$ 0.0
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K162500

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Product Description

Catalogue NumberK162500
Chemical NameKenpaullone
Synonyms9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one; 9-Bromopaullone; NSC 664704;
CAS Number142273-20-9
Molecular FormulaC₁₆H₁₁BrN₂O
AppearanceDark Yellow to Very Dark Yellow Solid
Melting Point>300°C
Molecular Weight327.18
Storage-20°C Freezer
SolubilityDMSO (Slightly), Methanol (Slightly, Heated)
Category Research Tools; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
ApplicationsThe paullones are a novel class of kinase inhibitors, initially identified as CDK inhibitors. Kenpaullone has been found to be a useful GSK-3ß inhibitor (IC50=23nM).
ReferencesZaharevitz, D.W., et al.: Cancer Res., 59, 2566 (1999), Leclerc, S., et al.: J. Biol. Chem., 276, 251 (2001), Bain, J., et al.: Biochem. J., in press.