G601510 Chemical Structure

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10mg
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50mg
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mg100
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  • Ships On : 7/12/2022
G601510

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Product Description

Catalogue NumberG601510
Chemical NameGDC-0941
Synonyms2-(1H-indazol-4-yl)-6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinothieno[3,2-d]pyrimidine; 4-[2-(1H-Indazol-4-yl)-6-[[4-(methylsulfonyl)piperazin-1-yl]methyl]thieno[3,2-d]pyrimidin-4-yl]morpholine; GDC 0941; GDC 941; GNE 0941; Pictilisib; Pictrelisib
CAS Number957054-30-7
Molecular Formula C23H27N7O3S2
AppearanceWhite to Off-White Solid
Melting Point>200ºC (dec.)
Molecular Weight513.64
Storage-20°C Freezer
SolubilityDMSO (Slightly), Methanol (Slightly, Heated)
Category Research Tools; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
ApplicationsGDC-0941 is a potent and selective oral inhibitor of the class I PI3K. GDC-0941 demonstrated broad spectrum of activity in breast, ovarian, lung, and prostate cancer models. Studies has also shown GDC-0941 may enhance anti-tumor activity of Docetaxel (D494420) in human breast cancer models. Potent PI3K inhibitor.
ReferencesJeffrey J.W., et al.: Clinical. Cancer. Rsch., 10, 1078 (2012); Murray, J.M., et al.: J. Medn. Chem., 55, 7686 (2012);