All Products are stable to be shipped at room temperature, unless otherwise specified.
Pack SizeQuantityPrice (USD)Sub Total
$ 1760.000.0
Exact Weight Packaging
$ 75.00 / Vial 0.0
Total$ 0.0
Request another packsize ? Click here.

Inventory Status : Currently Back Ordered - Please Request Lead Time

Bulk Order Request for T549002

#Pack SizeUnitQuantity

Product Description

Catalogue Number:T549002
Chemical Name:Tosedostat-d5
Synonyms:(αS)-α-[[(2R)-2-[(1S)-1-Hydroxy-2-(hydroxyamino)-2-oxoethyl]-4-methyl-1-oxopentyl]amino]benzeneacetic Acid-d5 Cyclopentyl Ester; CHR 2797-d5;
CAS Number:1217844-03-5
Alternate CAS #:unlabelled: 238750-77-1
Molecular Formula:C₂₁H₂₅D₅N₂O₆
Molecular Weight:411.5
Category: Standards; Isotopic Labeled Analogues; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
Applications:Labelled Tosedostat. CHR-2797 is a novel metalloenzyme inhibitor that is converted into a pharmacological active acid product (CHR-79888) inside cells. CHR-2797 exerts antiproliferative effects against a range of tumor cell lines in vitro and in vivo and shows selectivity for transformed over nontransformed cells. Its antiproliferative effects are at least 300 times more potent than the prototypical aminopeptidase inhibitor, Bestatin.