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Pack Size Quantity Price (USD) Sub Total
1mg
$ 115.00 0.0
2mg
$ 120.00 0.0
5mg
$ 130.00 0.0
10mg
$ 255.00 0.0
25mg
$ 500.00 0.0
50mg
$ 945.00 0.0
Exact Weight Packaging
$ 75.00 / Vial 0.0
Total $ 0.0
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Product Description

Catalogue Number: G797800
Chemical Name: GSK PERK Inhibitor
Synonyms: 1-[5-(4-Amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1H-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanone; 3-Fluoro-GSK2606414
CAS Number: 1337531-89-1
Molecular Formula: C₂₄H₁₉F₄N₅O
Appearance: Off-White to Pale Yellow Solid
Melting Point: 233-238°C (dec.)
Molecular Weight: 469.43
Storage: Refrigerator
Solubility: DMSO (Slightly), Methanol (Slightly, Heated)
Category: Research Tools; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
Applications: GSK PERK Inhibitor is an inhibitor of PERK, an important transmembrane protein of endoplasmic reticulum (ER). GSK PERK Inhibitor can be useful in the treatment of cancer, ocular diseases, and diseases associated with activated unfolded protein response pathways. As a result, GSK PERK Inhibitor has potential use in the treatment of diseases such as Alzheimer's disease, stroke, Type 1 diabetes, Parkinson disease, Huntington's disease, amyotrophic lateral sclerosis, myocardial infarction, cardiovascular disease, atherosclerosis, and arrhythmias, and more specifically cancers of the breast, colon, pancreatic, and lung.
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