All Products are stable to be shipped at room temperature, unless otherwise specified.
Pack SizeQuantityPrice (USD)Sub Total
5mg
$ 105.000.0
10mg
$ 160.000.0
50mg
$ 415.000.0
100mg
$ 675.000.0
200mg
$ 1040.000.0
Exact Weight Packaging
$ 75.00 / Vial 0.0
Total$ 0.0
Request another packsize ? Click here.

Inventory Status : In Stock

Bulk Order Request for C781800

#Pack SizeUnitQuantity
1.
2.
3.
4.
5.

Product Description

Catalogue Number:C781800
Chemical Name:Crenolanib Trifluoroacetic Acid Salt
Synonyms:1-[2-[5-[(3-Methyl-3-oxetanyl)methoxy]-1H-benzimidazol-1-yl]-8-quinolinyl]-4-piperidinamine Trifluoroacetic Acid Salt; ARO 002 Trifluoroacetic Acid Salt; CP 868596 Trifluoroacetic Acid Salt; [1-[2-[5-(3-Methyloxetan-3-ylmethoxy)benzimidazol-1-yl]quinolin-8-yl]piperidin-4-yl]amine Trifluoroacetic Acid Salt;
CAS Number:1797008-57-1
Alternate CAS #:Free amine: 670220-88-9
Molecular Formula:C₂₈H₃₀F₃N₅O₄
Appearance:Off-White to Pale Yellow Solid
Melting Point:214-217°C
Molecular Weight:557.56
Storage:Refrigerator
Solubility:DMSO (Slightly), Methanol (Very Slightly)
Category: Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
Applications:Crenolanib (CP-868569) is a tyrosine kinase inhibitor that acts by specifically inhibiting the receptor tyrosine kinases PDGFRα and PDGFRβ. Crenolanib (CP-868569) inhibits the activity of PDGFRα D842V kinase and prevented the phosphorylation of wild type PDGFRα. Crenolanib (CP-868569) possesses potential antineoplastic activity. Crenolanib is believed to suppress PDGFR-related signal transduction pathways leading to the inhibition of tumor angiogenesis and tumor cell proliferation.
References