Bromodomain Inhibitors

Bromodomain Inhibitors

Bromodomain Inhibitors are a class of antiviral drugs commonly used in the treatment of HIV. These molecules bind to regions of proteins known as bromodomains— which bind acetylated lysines in histone tails. Proteins that contain bromodomains are also epigenetic regulators, which play an important role in gene expression and regulation. This class of inhibitors blocks these protein interactions and in turn prevents viral replication within the host cell.

Discover our complete range of inhibitors and modulators along with building blocks, metabolites, impurities and labelled isotopes.

Displaying 0 - 12 of 27 Results

2-Methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide

 2-Methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide
  • Catalogue NumberM264535
  • CAS1403764-72-6
  • Molecular FormulaC₁₆H₁₇N₃O₄S

I-BET 151

 I-BET 151
  • Catalogue NumberI120050
  • CAS1300031-49-5
  • Molecular FormulaC₂₃H₂₁N₅O₃

(S)-(+)-Tert-butyl 2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetate

 (S)-(+)-Tert-butyl 2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetate
  • Catalogue NumberT117580
  • CAS1268524-70-4
  • Molecular FormulaC₂₃H₂₅ClN₄O₂S

Controlled Substance

 Controlled Substance
  • Catalogue NumberC375140
  • ----
  • ----

SGC-CBP30

 SGC-CBP30
  • Catalogue NumberS282310
  • CAS1613695-14-9
  • Molecular FormulaC₇H₁₀N₂O₄

I-CBP 112 Hydrochloride Salt

 I-CBP 112 Hydrochloride Salt
  • Catalogue NumberI163880
  • CAS2147701-33-3
  • Molecular FormulaC₂₇H₃₆N₂O₅• HCl

Bromosporine

 Bromosporine
  • Catalogue NumberB687500
  • CAS1619994-69-2
  • Molecular FormulaC₁₇H₂₀N₆O₄S

Controlled Substance

 Controlled Substance
  • Catalogue NumberC781425
  • ----
  • ----

4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methylbenzenesulfonamide

 4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methylbenzenesulfonamide
  • Catalogue NumberB683530
  • CAS919973-83-4
  • Molecular FormulaC₁₇H₁₈BrN₃O₄S

3-Formylphenylboronic Acid

 3-Formylphenylboronic Acid
  • Catalogue NumberF700970
  • CAS87199-16-4
  • Molecular FormulaC₇H₇BO₃

4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methylbenzenesulfonamide-d6

 4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methylbenzenesulfonamide-d6
  • Catalogue NumberB683532
  • CAS---
  • Molecular FormulaC₁₇H₁₂D₆BrN₃O₄S

4-Cyanobenzaldehyde

 4-Cyanobenzaldehyde
  • Catalogue NumberC962305
  • CAS105-07-7
  • Molecular FormulaC₈H₅NO