Bromodomain Inhibitors

Bromodomain Inhibitors are a class of antiviral drugs commonly used in the treatment of HIV. These molecules bind to regions of proteins known as bromodomains— which bind acetylated lysines in histone tails. Proteins that contain bromodomains are also epigenetic regulators, which play an important role in gene expression and regulation. This class of inhibitors blocks these protein interactions and in turn prevents viral replication within the host cell.

Discover our complete range of inhibitors and modulators along with building blocks, metabolites, impurities and labelled isotopes.

Displaying 0 - 12 of 34 Results

2-Methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide

2-Methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide
  • Catalogue NumberM264535
  • CAS1403764-72-6
  • Molecular FormulaC₁₆H₁₇N₃O₄S

I-BET 151

I-BET 151
  • Catalogue NumberI120050
  • CAS1300031-49-5
  • Molecular FormulaC₂₃H₂₁N₅O₃

SGC-CBP30

SGC-CBP30
  • Catalogue NumberS282310
  • CAS1613695-14-9
  • Molecular FormulaC₂₈H₃₃ClN₄O₃

I-CBP 112 Hydrochloride Salt

I-CBP 112 Hydrochloride Salt
  • Catalogue NumberI163880
  • CAS2147701-33-3
  • Molecular FormulaC₂₇H₃₆N₂O₅• HCl

Bromosporine

Bromosporine
  • Catalogue NumberB687500
  • CAS1619994-69-2
  • Molecular FormulaC₁₇H₂₀N₆O₄S

CPI-203

CPI-203
  • Catalogue NumberC781425
  • CAS1446144-04-2
  • Molecular FormulaC₁₉H₁₈ClN₅OS

4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methylbenzenesulfonamide

4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methylbenzenesulfonamide
  • Catalogue NumberB683530
  • CAS919973-83-4
  • Molecular FormulaC₁₇H₁₈BrN₃O₄S

3-Formylphenylboronic Acid

3-Formylphenylboronic Acid
  • Catalogue NumberF700970
  • CAS87199-16-4
  • Molecular FormulaC₇H₇BO₃

4-Cyanobenzaldehyde

4-Cyanobenzaldehyde
  • Catalogue NumberC962305
  • CAS105-07-7
  • Molecular FormulaC₈H₅NO