Sumanirole Maleate

Catalogue number: S790700
Chemical name: Sumanirole Maleate
Synonyms: (5R)-5,6-Dihydro-5-(methylamino)-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (2Z)-2-Butenedioate; (R)-5,6-Dihydro-5-(methylamino)-4H-imidazo[4,5,1-ij]quinolin- 2(1H)-one (2Z)-2-Butenedioate;
CAS Number: 179386-43-7
Possible CAS #: NA
Molecular form.: C₁₅H₁₇N₃O₅
Appearance: Off-White to Light Beige Solid
Melting Point: 200-208°C (dec.)
Mol. Weight: 319.31
Storage: Refrigerator
Solubility: DMSO, Methanol
Stability: No Data Available
Category: Amines, Aromatics, Chiral Reagents, Pfizer compounds, Pharmaceuticals, Intermediates & Fine Chemicals,
Boiling Point: No Data Available
Applications: Sumanirole is a high affinity D2 receptor agonist (EC50 values are between 17 and 75 nM in cell-based assays). Sumanirole displays >200-fold selectivity for the D2 receptor against other dopamine receptor subtypes (Ki values are 9.0, 1940, >2190 and >7140 for D2, D3, D4 and D1 receptors respectively). Sumanirole exhibits antiParkinsonian activity similar to Ropinirole (R641000).
Dangerous Goods Info: NA
References:
Peer Review Product Citations:

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