SB 242084

Catalogue number: S154450
Chemical name: SB 242084
Synonyms: 6-Chloro-2,3-dihydro-5-methyl-N-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-1H-indole-1-carboxamide;
CAS Number: 181632-25-7
Possible CAS #: NA
Molecular form.: C₂₁H₁₉ClN₄O₂
Appearance: Off-White Solid
Melting Point: 176-178°C
Mol. Weight: 394.85
Storage: Refrigerator
Solubility: Methanol
Stability: No Data Available
Category: Amines, Aromatics, Heterocycles, Pharmaceuticals, Intermediates & Fine Chemicals
Boiling Point: No Data Available
Applications: SB 242084 is a 5-HT2C receptor antagonist that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively. SB 242084 displays selectivity over a range of other 5-HT, dopamine and adrenergic receptors.SB 242084 os a brain penetrant; exerts anxiolytic-like activity.
Dangerous Goods Info: NA
References: Bromidge, et al.: J. Med. Chem., 40, 3494 (1997), Kennet, et al.: Neuropharmacology, 36, 609 (1997), Dalton, et al.: Psychopharmacology, 185, 45 (2006),
Peer Review Product Citations:

Order Product

  Pack size Price(USD)
10mg $150.00
  Pack size Price(USD)
100mg $1200.00
Exact Weight Packaging ($75(USD) / Vial)
Inventory Status:   Pending QC

Search Products:

Enter Catalogue #, CAS # , Chemical Name or Mol Formula:

Search By Category

Search By Category View products by category
Translate »