Loperamide-d6 N-Oxide

Catalogue number: L469462
Chemical name: Loperamide-d6 N-Oxide
Synonyms: trans-4-(4-Chlorophenyl)-4-hydroxy-N,N-(dimethyl-d6)-α,α-diphenyl-1-piperidinebutanamide 1-Oxide; Arestal-d6; Loperamide-d6 Oxide; R 58425-d6;
CAS Number: 1329835-39-3
Possible CAS #: unlabelled: 106900-12-3
Molecular form.: C₂₉H₂₇D₆ClN₂O₃
Appearance: No Data Available
Melting Point: No Data Available
Mol. Weight: 499.07
Storage: No Data Available
Solubility: No Data Available
Stability: No Data Available
Category: Drug Analogues, Heterocycles, Isotope Labelled Compounds, Metabolites & Impurities, Pharmaceuticals, Intermediates & Fine Chemicals,
Boiling Point: No Data Available
Applications: Labelled Loperamide oxide (LOPOX). It is a prodrug of Loperamide (LOP). It is concluded that Loperamide oxide administered intraluminally is reduced to Loperamide and has the same antisecretory potency as Loperamide in jejunum and colon.
Dangerous Goods Info: NA
References: Lavrijsen, K., et al.: Drug Metab. Dispos., 23, 354 (1995), Hesselink, D., et al.: Clin. Pharmacol. Ther., 74, 245 (2003), Hooijberg, J., et al.: Biochem. Pharmacol., 67, 1541 (2004),
Peer Review Product Citations:

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