Catalogue number: K162500
Chemical name: Kenpaullone
Synonyms: 9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one; 9-Bromopaullone; NSC 664704;
CAS Number: 142273-20-9
Possible CAS #: NA
Molecular form.: C₁₆H₁₁BrN₂O
Appearance: Dark Yellow to Very Dark Yellow Solid
Melting Point: >300°C
Mol. Weight: 327.18
Storage: -20°C Freezer
Solubility: DMSO (Slightly), Methanol (Slightly, Heated)
Stability: No Data Available
Category: Aromatics, Heterocycles, Inhibitors, Pharmaceuticals, Intermediates & Fine Chemicals
Boiling Point: No Data Available
Applications: The paullones are a novel class of kinase inhibitors, initially identified as CDK inhibitors. Kenpaullone has been found to be a useful GSK-3ß inhibitor (IC50=23nM).
References: Zaharevitz, D.W., et al.: Cancer Res., 59, 2566 (1999), Leclerc, S., et al.: J. Biol. Chem., 276, 251 (2001), Bain, J., et al.: Biochem. J., in press.
Dangerous Goods Info: NA

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  Pack size Price(USD)
1mg $45.00
10mg $120.00
50mg $550.00
  Pack size Price(USD)
5mg $85.00
25mg $290.00
100mg $960.00
Exact Weight Packaging ($75(USD) / Vial)
Inventory Status:   In Stock

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