GSK PERK Inhibitor-d3

Catalogue number: G797802
Chemical name: GSK PERK Inhibitor-d3
Synonyms: 1-[5-(4-Amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1H-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanone-d3; 3-Fluoro-GSK2606414-d3
CAS Number: NA
Possible CAS #: Unlabelled: 1337531-89-1
Molecular form.: C₂₄H₁₆D₃F₄N₅O
Appearance: No Data Available
Melting Point: No Data Available
Mol. Weight: 472.45
Storage: No Data Available
Solubility: No Data Available
Stability: No Data Available
Category: Aromatics, Heterocycles, Indole Derivatives, Inhibitors, Isotope Labelled Compounds, Pharmaceuticals, Intermediates & Fine Chemicals,
Boiling Point: No Data Available
Applications: Labelled GSK PERK Inhibitor is an inhibitors of PERK, an important transmembrane protein of endoplasmic reticulum (ER). GSK PERK Inhibitor can be useful in the treatment of cancer, ocular diseases, and diseases associated with activated unfolded protein response pathways. As a result, GSK PERK Inhibitor has potential use in the treatment of diseases such as Alzheimer’s disease, stroke, Type 1 diabetes, Parkinson disease, Huntington’s disease, amyotrophic lateral sclerosis, myocardial infarction, cardiovascular disease, atherosclerosis, and arrhythmias, and more specifically cancers of the breast, colon, pancreatic, and lung.
References: Baltzis, D. et al.: J. Biol. Chem., 282, 31675 (2007); Axten, J. al,: J. Med. Chem. 55(16) 7193 (2012).
Dangerous Goods Info: NA

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  Pack size Price(USD)
1mg $225.00
  Pack size Price(USD)
10mg $1800.00
Exact Weight Packaging ($75(USD) / Vial)
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