Catalogue number: G797600
Chemical name: GSK360A
Synonyms: N-[[1-(2-Cyclopropylethyl)-6-fluoro-1,2-dihydro-4-hydroxy-2-oxo-3-quinolinyl]carbonyl]glycine; N-[[1-(2-Cyclopropylethyl)-6-fluoro-4-hydroxy-2-oxo-1,2-dihydro-3-quinolinyl]carbonyl]glycine;
CAS Number: 931399-19-8
Possible CAS #: 680590
Molecular form.: C₁₇H₁₇FN₂O₅
Appearance: Beige Solid
Melting Point: 194-198°C (dec.)
Mol. Weight: 348.33
Storage: Refrigerator
Solubility: DMSO, Methanol
Stability: No Data Available
Category: Aromatics, Heterocycles, Inhibitors, Pharmaceuticals, Intermediates & Fine Chemicals,
Boiling Point: No Data Available
Applications: GSK360A orally active HIF-PHD inhibitor. GSK360A exerts systemic and local effects by stabilizing HIF-1α signaling and improves long-term ventricular function, remodeling, and vascularity in a model of established ventricular dysfunction. These findings suggest that GSK360A may be suitable for the treatment of post-MI remodeling and heart failure.
Dangerous Goods Info: NA
References: Bao, W.-K. et al.: J. Cardio. Pharmacol., 56, 147 (2010);
Peer Review Product Citations: Bao, W.-K. et al.: J. Cardio. Pharmacol., 56, 147 (2010);

Order Product

  Pack size Price(USD)
2mg $110.00
10mg $285.00
50mg $1200.00
  Pack size Price(USD)
5mg $150.00
25mg $700.00
Exact Weight Packaging ($75(USD) / Vial)
Inventory Status:   In Stock

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