Esterastin DISCONTINUED

Catalogue number: E668400
Chemical name: Esterastin DISCONTINUED
Synonyms: N2-Acetyl-L-asparagine (1S,3Z,6Z)-1-[[(2S,3S)-3-Hexyl-4-oxo-2-oxetanyl] methyl]-3,6-dodecadien-1-yl Ester; [2S-[2α(1R*,3Z,6Z),3β]]-N2-Acetyl-L-asparagine 1-[(3-Hexyl-4-oxo-2-oxetanyl) methyl]-3,6-dodecadienyl Ester;
CAS Number: 67655-93-0
Possible CAS #: NA
Molecular form.: C₂₈H₄₆N₂O₆
Appearance: No Data Available
Melting Point: No Data Available
Mol. Weight: 506.67
Storage: Amber Vial, -20°C Freezer, Under inert atmosphere
Solubility: No Data Available
Stability: No Data Available
Category: Amino Acids & Derivatives, Chiral Reagents, Heterocycles, Pharmaceuticals, Intermediates & Fine Chemicals
Boiling Point: No Data Available
Applications: Esterastin is a potent inhibitor of lysosomal acid lipase. Esterastin inhibited the enzyme activity very strongly (IC50, about 80 nM). The inhibition of acid lipase by Esterastin was competitive with respect to the substrate and the inhibition constant for Esterastin was 90 nM. Esterastin was less inhibitory to other lipolytic enzymes, such as pancreatic lipase and carboxylesterase. Thus, Esterastin is a potent new inhibitor of lysosomal acid lipase.
Dangerous Goods Info: NA
References:
Peer Review Product Citations:

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