CP 945598 Hydrochloride

Catalogue number: C781420
Chemical name: CP 945598 Hydrochloride
Synonyms: 1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-4-(ethylamino)-4-piperidinecarboxamide Hydrochloride; 1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]- 4-(ethylamino)-4-piperidinecarboxamide Monohydrochloride; CP 945598; CP 945598-01; Otenabant Hydrochloride;
CAS Number: 686347-12-6
Possible CAS #: 686344-29-6-free base
Molecular form.: C₂₅H₂₆Cl₃N₇O
Appearance: Off-White Solid
Melting Point: 283-291°C
Mol. Weight: 546.88
Storage: Refrigerator
Solubility: DMSO (Sparingly), Methanol (Sparingly)
Stability: No Data Available
Category: Amines, Aromatics, Heterocycles, Pfizer Compounds, Pharmaceuticals, Intermediates & Fine Chemicals
Boiling Point: No Data Available
Applications: CP 945598 is a selective, high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional assays respectively). Displays low affinity for CB2 receptors (Ki = 7600 nM).
Dangerous Goods Info: NA
References: Griffith, et al.: J. Med. Chem., 52, 234 (2009), Hadcock, et al.: Biochem. Biophys. Res. Commun., 394, 366 (2010),
Peer Review Product Citations:

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  Pack size Price(USD)
5mg $75.00
25mg $175.00
250mg $975.00
  Pack size Price(USD)
10mg $95.00
100mg $475.00
500mg $1750.00
Exact Weight Packaging ($75(USD) / Vial)
Inventory Status:   Pending QC

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