CP-100356 Hydrochloride

Catalogue number: C781250
Chemical name: CP-100356 Hydrochloride
Synonyms: 4-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-6,7-dimethoxy-2-quinazolinamine Monohydrochloride;
CAS Number: 142715-48-8
Possible CAS #: NA
Molecular form.: C₃₁H₃₇ClN₄O₆
Appearance: Off-White to Light Tan Solid
Melting Point: 210-212°C
Mol. Weight: 597.1
Storage: Refrigerator
Solubility: Chloroform, Methanol
Stability: No Data Available
Category: Amine, Aromatics, Heterocycles, Pfizer Compounds, Pharmaceuticals, Intermediates & Fine Chemicals
Boiling Point: No Data Available
Applications: CP-100356 is a specific inhibitor of MDR1 (P-Gp), the protypical ABC transporter. CP-100356 also inhibits prazosin transport in human breast cancer resistance protein (BCRP)-transfected MDCKII cells, suggesting that it acts as a dual inhibitor. CP-100356 does not inhibit multidrug resistance-associated protein 2 (MPR2 IC50 >15 mM).
Dangerous Goods Info: NA
References:
Peer Review Product Citations:

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100mg $1280.00
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Exact Weight Packaging ($75(USD) / Vial)
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Inventory Status:   Pending QC

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