Aprepitant

Catalogue number: A729800
Chemical name: Aprepitant
Synonyms: 5-[[(2R,3S)-2-[(1R)-1-[3,5-Bis(trifluoromethyl)phenyl]ethoxy]-3-(4-fluorophenyl)-4-morpholinyl]methyl]-1,2-dihydro-3H-1,2,4-triazol-3-one; Emend; L 754030; MK 0869; MK 869; ONO 7436;
CAS Number: 170729-80-3
Possible CAS #: NA
Molecular form.: C₂₃H₂₁F₇N₄O₃
Appearance: White to Pale Beige Solid
Melting Point: 242-250°C
Mol. Weight: 534.43
Storage: -20°C Freezer
Solubility: DMSO, Methanol
Stability: No Data Available
Category: Chiral Reagents, Heterocycles, Pharmaceuticals, Intermediates & Fine Chemicals,
Boiling Point: No Data Available
Applications: A novel selective neurokinin-1 (NK-1) receptor antagonist. In vitro studies using human liver microsomes indicate that Aprepitant is metabolised primarily by CYP3A4 with minor metabolism by CYP1A2 and CYP2C19, and no metabolism by CYP2D6, CYP2C9, or CYP2E1. Antiemetic.
Dangerous Goods Info: NA
References:
Peer Review Product Citations:

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25mg $150.00
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250mg $425.00
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